Compile Data Set for Download or QSAR
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Found 235 from University of Southampton
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083326(3-Acetylamino-6-dihydroxymethyl-4-guanidino-3,4-di...)
Affinity DataKi:  0.130nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083322(3-Acetylamino-2-diethylcarbamoyl-6-dihydroxymethyl...)
Affinity DataKi:  0.390nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083320(3-Acetylamino-6-dihydroxymethyl-2-(phenethyl-propy...)
Affinity DataKi:  0.650nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083327(3-Acetylamino-6-dihydroxymethyl-4-guanidino-3,4-di...)
Affinity DataKi:  0.650nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083333(CHEMBL348207 | N-[6-Dihydroxymethyl-4-guanidino-2-...)
Affinity DataKi:  1nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50399614(CHEMBL2181170)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083328(3-Acetylamino-6-dihydroxymethyl-4-guanidino-3,4-di...)
Affinity DataKi:  3.30nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50443687(CHEMBL3093187)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50443688(CHEMBL3093186)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50443690(CHEMBL3093184)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50399619(CHEMBL2181189)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50443691(CHEMBL3093194)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083324((2R,3R,4S)-3-Acetylamino-6-dihydroxymethyl-2-((R)-...)
Affinity DataKi:  40nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50399632(CHEMBL2177145)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50443689(CHEMBL3093185)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083332((2R,3R,4R)-3-Acetylamino-6-dihydroxymethyl-2-((R)-...)
Affinity DataKi:  100nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083325(3-Acetylamino-6-dihydroxymethyl-2-dimethylcarbamoy...)
Affinity DataKi:  310nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional purine biosynthesis protein ATIC(Homo sapiens (Human))
University of Southampton

LigandPNGBDBM92374(RY Analogue, 14)
Affinity DataKi:  685nM ΔG°:  -8.40kcal/moleT: 2°CAssay Description:Enzyme inhibition using aminoimidazole carboxamide ribonucleotide transformylase/inosine monophosphate cyclohydrolase (ATIC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083331(3-Acetylamino-6-dihydroxymethyl-4-guanidino-3,4-di...)
Affinity DataKi:  910nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50443688(CHEMBL3093186)
Affinity DataKi:  1.20E+3nMAssay Description:Binding affinity to human 5HT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083319(3-Acetylamino-6-dihydroxymethyl-2-phenethylcarbamo...)
Affinity DataKi:  1.57E+3nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083321(3-Acetylamino-6-dihydroxymethyl-2-ethylcarbamoyl-3...)
Affinity DataKi:  1.69E+3nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50346584(CHEMBL1795979)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50346585(CHEMBL1795980 | S2101)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50346586(CHEMBL1795981 | US8765820, 5a)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional purine biosynthesis protein ATIC(Homo sapiens (Human))
University of Southampton

LigandPNGBDBM92376(RY Analogue, 17)
Affinity DataKi:  2.50E+3nM ΔG°:  -7.64kcal/moleT: 2°CAssay Description:Enzyme inhibition using aminoimidazole carboxamide ribonucleotide transformylase/inosine monophosphate cyclohydrolase (ATIC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50443687(CHEMBL3093187)
Affinity DataKi:  2.60E+3nMAssay Description:Binding affinity to human 5HT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCatenin beta-1(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50014132(CHEMBL2323032)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity to beta catenin ARD (142 to 686 residues) (unknown origin) assessed as inhibition constant by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50371232(CARNOSIC ACID)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity to N-terminal FLAG tagged beta catenin (134 to 671 residues)/FLAG tagged BCL9 domain 2 (343 to 396 residues) (unknown origin) protei...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50346589(CHEMBL1795974 | CHEMBL255520)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083323(CHEMBL148966 | N-[(2R,3R,4S)-6-Dihydroxymethyl-4-h...)
Affinity DataKi:  4.00E+3nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50346583(CHEMBL1795978)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50346591(CHEMBL1795982)
Affinity DataKi:  6.80E+3nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50346582(CHEMBL1795977)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50346590(CHEMBL1795975)
Affinity DataKi:  8.90E+3nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083329(CHEMBL147080 | [(2R,3R,4S)-3-Acetylamino-6-dihydro...)
Affinity DataKi:  1.00E+4nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50346594(CHEMBL1795976)
Affinity DataKi:  1.17E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-(-)-2-phenylcyclopropylamine | (1R,2S)-2-p...)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50083330(3-Acetylamino-6-dihydroxymethyl-2-methylcarbamoyl-...)
Affinity DataKi:  2.40E+4nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50113851((+/-)-Tranylcypromine | 2-PCPA | 2-Phenyl-cyclopro...)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | CHEMBL25799...)
Affinity DataKi:  2.66E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | CHEMBL25799...)
Affinity DataKi:  2.81E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50346587(CHEMBL1795972)
Affinity DataKi:  4.18E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional purine biosynthesis protein ATIC(Homo sapiens (Human))
University of Southampton

LigandPNGBDBM92372(RY Analogue, 12)
Affinity DataKi:  5.60E+4nM ΔG°:  -5.80kcal/moleT: 2°CAssay Description:Enzyme inhibition using aminoimidazole carboxamide ribonucleotide transformylase/inosine monophosphate cyclohydrolase (ATIC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional purine biosynthesis protein ATIC(Homo sapiens (Human))
University of Southampton

LigandPNGBDBM92373(RY Analogue, 13)
Affinity DataKi:  5.90E+4nM ΔG°:  -5.77kcal/moleT: 2°CAssay Description:Enzyme inhibition using aminoimidazole carboxamide ribonucleotide transformylase/inosine monophosphate cyclohydrolase (ATIC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50346588(CHEMBL1795973)
Affinity DataKi:  7.96E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional purine biosynthesis protein ATIC(Homo sapiens (Human))
University of Southampton

LigandPNGBDBM92368(RY Analogue, 8)
Affinity DataKi:  8.40E+4nM ΔG°:  -5.56kcal/moleT: 2°CAssay Description:Enzyme inhibition using aminoimidazole carboxamide ribonucleotide transformylase/inosine monophosphate cyclohydrolase (ATIC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional purine biosynthesis protein ATIC(Homo sapiens (Human))
University of Southampton

LigandPNGBDBM92371(RY Analogue, 11)
Affinity DataKi:  8.70E+4nM ΔG°:  -5.54kcal/moleT: 2°CAssay Description:Enzyme inhibition using aminoimidazole carboxamide ribonucleotide transformylase/inosine monophosphate cyclohydrolase (ATIC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50346592(CHEMBL1795983)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50346593(CHEMBL1795984)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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