TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 0.390nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 0.650nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 0.650nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
Affinity DataKi: 685nM ΔG°: -8.40kcal/moleT: 2°CAssay Description:Enzyme inhibition using aminoimidazole carboxamide ribonucleotide transformylase/inosine monophosphate cyclohydrolase (ATIC).More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 910nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity to human 5HT3More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 1.57E+3nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 1.69E+3nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nM ΔG°: -7.64kcal/moleT: 2°CAssay Description:Enzyme inhibition using aminoimidazole carboxamide ribonucleotide transformylase/inosine monophosphate cyclohydrolase (ATIC).More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:Binding affinity to human 5HT3More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity to beta catenin ARD (142 to 686 residues) (unknown origin) assessed as inhibition constant by fluorescence polarisation assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity to N-terminal FLAG tagged beta catenin (134 to 671 residues)/FLAG tagged BCL9 domain 2 (343 to 396 residues) (unknown origin) protei...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 3.70E+3nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 4.00E+3nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 6.80E+3nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 8.90E+3nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 1.17E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 2.10E+4nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 2.40E+4nMAssay Description:Neuraminidase binding affinity in Influenza AMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 2.50E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 2.66E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 2.81E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 4.18E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
Affinity DataKi: 5.60E+4nM ΔG°: -5.80kcal/moleT: 2°CAssay Description:Enzyme inhibition using aminoimidazole carboxamide ribonucleotide transformylase/inosine monophosphate cyclohydrolase (ATIC).More data for this Ligand-Target Pair
Affinity DataKi: 5.90E+4nM ΔG°: -5.77kcal/moleT: 2°CAssay Description:Enzyme inhibition using aminoimidazole carboxamide ribonucleotide transformylase/inosine monophosphate cyclohydrolase (ATIC).More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: 7.96E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
Affinity DataKi: 8.40E+4nM ΔG°: -5.56kcal/moleT: 2°CAssay Description:Enzyme inhibition using aminoimidazole carboxamide ribonucleotide transformylase/inosine monophosphate cyclohydrolase (ATIC).More data for this Ligand-Target Pair
Affinity DataKi: 8.70E+4nM ΔG°: -5.54kcal/moleT: 2°CAssay Description:Enzyme inhibition using aminoimidazole carboxamide ribonucleotide transformylase/inosine monophosphate cyclohydrolase (ATIC).More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair